Acute myeloid leukaemias (AMLs) have a low mutational burden compared to other cancers. Familial cases of AML are rare and often have pre-existing myelodysplastic or bone marrow failure syndromes. Base excision repair proteins (BER) like MBD4 have been linked to solid cancers but not haematological malignancies.
Three patients, of whom 2 are siblings, with no previous haematological disorders, developed AML at a young age (<35 years old). All patients had complete loss of MBD4 through germline loss of function mutations. The AMLs were characterised by a high somatic mutation rate (~33 fold above a typical AML). More than 95% of somatic mutations were cytosine to thymine (C>T) mutations in the context of a methylated CG dinucleotide (CG>TG mutations).
The AMLs had a distinctive mutational signature, akin to an extreme form of Signature 1. Nine cancers out of 10,638 in the TCGA database also had MBD4 mutations. In a uveal melanoma and a glioblastoma multiforme, the wild type MBD4 allele was lost through copy number alterations. These 2 cancers also had a high mutation rate and the same extreme Signature 1 as our AMLs. Whole genome sequencing of individual myeloid progenitor colonies of MBD4+/+ and MBD4-/- mice recapitulated the high mutation rate and Signature 1. This is consistent with constant deamination of methylcytosine (5mC) in cells, resulting in C>T mutations, and is usually repaired by MBD4.
Our AMLs had somatic mutations in the same genes, acquired in the same order (biallelic DNMT3A mutations followed by IDH1/2 mutations). We propose that loss of MBD4 impairs repair of C>T mutations, accelerating the clock-like mutational process of Signature 1. In the haematopoietic compartment, acquisition of DNMT3A mutations provides a selective advantage for that clone. Additional mutations in IDH1/2 and other genes due to impaired BER ultimately result in AML. Furthermore, discovery of other cancers with acquired loss of MBD4 and the same distinctive mutational signature suggests a role in other malignancies.